CC-115 hydrochloride
Cat. No.:YN420248
| 产品名称: | CC-115 hydrochloride |
| CAS No.: | 1300118-55-1 |
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| 分子量: | 372.81 |
| 分子式: | C₁₆H₁₇ClN₈O |
| SMILES: | [H]Cl.O=C1CN=C2C(N1CC)=NC(C3=C(C)N=C(C4=NN=CN4)C=C3)=CN2 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | CC-115 hydrochloride 是一种有效的双重DNA-PK和mTOR抑制剂,IC50分别为 13 nM 和 21 nM。CC-115 阻断mTORC1和mTORC2信号通路。 |
| IC50和靶点: | [{name:"DNA-PK:13 nM (IC50)"},{name: "mTOR:21 nM (IC50)'}, 'mTORC1', 'mTORC2', {'PI3Kα:852 nM (IC50)"}] |
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