FN-1501
Cat. No.:YN440144
| 产品名称: | FN-1501 |
| CAS No.: | 1429515-59-2 |
| Chemical Name: | |
| Synonyms: | |
| 分子量: | 431.49 |
| 分子式: | C₂₂H₂₅N₉O |
| SMILES: | O=C(C1=NNC=C1NC2=NC=NC3=C2C=CN3)NC4=CC=C(CN5CCN(C)CC5)C=C4 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | FN-1501 是一种有效的FLT3和CDK抑制剂,对 CDK2/cyclin A,CDK4/cyclin D1,CDK6/cyclin D1 和 FLT3 的IC50值分别为 2.47,0.85,1.96, 和 0.28 nM。FN-1501 具有抗肿瘤的活性。 |
| IC50和靶点: | [{name:"Cdk4/cyclin D1:0.85 nM (IC50)"},{name: "CDK6/cyclinD1:1.96 nM (IC50)"},{name: "cdk2/cyclin A:2.47 nM (IC50)"},{name: "FLT3:0.28 nM (IC50)"}] |
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