DK419
Cat. No.:YN450042
| 产品名称: | DK419 |
| CAS No.: | 2102672-22-8 |
| Chemical Name: | |
| Synonyms: | DK-419;DK 419 |
| 分子量: | 407.70 |
| 分子式: | C₁₆H₈ClF₆N₃O |
| SMILES: | O=C(C1=C2C(N=C(C(F)(F)F)N2)=CC(Cl)=C1)NC3=CC=C(C(F)(F)F)C=C3 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | DK419 是一种有效、可口服的Wnt/β-catenin信号通路抑制剂,IC50值为 0.19 μM。DK419 能降低 Axin2,β-catenin,c-Myc,Cyclin D1 和 Survivin 能够改变细胞内耗氧率,诱导 pAMPK 的产生。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |