Hydroxyfasudil
Cat. No.:YN450086
| 产品名称: | Hydroxyfasudil |
| CAS No.: | 105628-72-6 |
| Chemical Name: | |
| Synonyms: | 羟基法舒地尔; HA-1100 |
| 分子量: | 307.37 |
| 分子式: | C₁₄H₁₇N₃O₃S |
| SMILES: | O=C1NC=CC2=C1C=CC=C2S(=O)(N3CCNCCC3)=O |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | Hydroxyfasudil 是一种ROCK抑制剂,可抑制ROCK1和ROCK2的活性,IC50值分别为 0.73 和 0.72 μM。 |
| IC50和靶点: | [{name:"ROCK2:0.72 μM (IC50)"},{name: "ROCK1:0.73 μM (IC50)"},{name: "PKA:37 μM (IC50)"}] |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |