GSK2798745
Cat. No.：YN360692
CAS No. ：1419609-94-1
| 产品名称: | GSK2798745 |
| CAS No.: | 1419609-94-1 |
| Chemical Name: | |
| Synonyms: | GSK2798745;GSK-2798745;GSK 2798745 |
| 分子量: | 460.53 |
| 分子式: | C₂₅H₂₈N₆O₃ |
| SMILES: | N#CC1=CC=C2N=CN(C[C@](CCC3)(C)C[C@@]43CN(C5=NC=C(C(C)(O)C)N=C5)C(O4)=O)C2=C1 |
| 存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
| 运输: | Room temperature in continental US; may vary elsewhere. |
| 产品描述: | GSK2798745 是首创的，高效的，选择性的且具有口服活性的 瞬时受体电位香草酸 4(TRPV4)离子通道阻断剂，对于 hTRPV4 和 rTRPV4 的IC50值分别为 1.8 和 1.6 nM。GSK2798745 用于充血性心力衰竭相关的肺水肿的研究。 |
| IC50和靶点: | |
| In Vitro: | |
| In Vivo: | |
| Clinical Trial: | |
| Solvent & Solubility: |
