MPEP
Cat. No.:YN320897
CAS No. :96206-92-7
产品名称: | MPEP |
CAS No.: | 96206-92-7 |
Chemical Name: | |
Synonyms: | |
分子量: | 193.24 |
分子式: | C₁₄H₁₁N |
SMILES: | CC1=NC(C#CC2=CC=CC=C2)=CC=C1 |
存储: | Please store the product under the recommended conditions in theCertificate of Analysis. |
运输: | Room temperature in continental US; may vary elsewhere. |
产品描述: | MPEP 是有效的、选择性的、非竞争性的、口服有效的、具有系统活性的mGlu5受体拮抗剂,其完全抑制quisqualate 刺激的磷酸肌醇水解的IC50值为 36 nM。MPEP 具有抗焦虑或抗抑郁活性。 |
IC50和靶点: | [{name:"mGluR5:36 nM (IC50)"}] |
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In Vivo: | |
Clinical Trial: | |
Solvent & Solubility: |